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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TOP1 21,22-O-Diangeloyl-3beta,16alpha,28-trihydroxyolean-12-ene NA 250000 NA NA NA NA TTD
TOP1 2,4-Pyrimidinediamine, 6-chloro-N4-(3,4-dichlorophenyl)- NA 200000 NA NA NA NA TTD
TOP1 Camptothecin NA 127000 NA NA NA NA PubChem
TOP1 [(3R,4S,5R)-3,4-dihydroxy-5-[5-hydroxy-2-(4-hydroxyphenyl)-4-oxo-7-[(2S,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxychromen-3-yl]oxyoxolan-3-yl]methyl acetate NA 150000 NA NA NA NA TTD
TOP1 Doxorubicin NA 200000 NA NA NA NA PubChem
TOP1 Etoposide NA 1000000 NA NA NA NA PubChem|TTD
TOP1 Ginsenoside B2 NA 250000 NA NA NA NA PubChem|TTD
TOP1 2,4,6-Tri-furan-2-yl-pyridine NA 500000 NA NA NA NA TTD
TOP1 4-Furan-2-yl-2-thiophen-2-yl-pyridine NA 400000 NA NA NA NA TTD
TOP1 6-(1-Hydroxy-propyl)-5,8-dimethoxy-[1,4]naphthoquinone NA 121830 NA NA NA NA TTD
TOP1 (3E)-3-[(4-fluorophenyl)methylidene]-1-benzofuran-2-one NA 392000 NA NA NA NA TTD
TOP1 ethyl 2-[4-[(E)-(2-oxo-1-benzofuran-3-ylidene)methyl]phenyl]acetate NA 1000000 NA NA NA NA TTD
TOP1 (3E)-3-[(4-hydroxyphenyl)methylidene]-1-benzofuran-2-one NA 250000 NA NA NA NA TTD
TOP1 (E)-3-(3,4-Dihydroxybenzylidene)benzofuran-2(3H)-one NA 160000 NA NA NA NA TTD
TOP1 (3E)-3-[(3-hydroxyphenyl)methylidene]-1-benzofuran-2-one NA 262000 NA NA NA NA TTD
TOP1 (3E)-3-benzylidene-5-hydroxy-1-benzofuran-2-one NA 960000 NA NA NA NA TTD
TOP1 (3E)-3-[(4-hydroxy-3-methoxyphenyl)methylidene]-1-benzofuran-2-one NA 630000 NA NA NA NA TTD
TOP1 Gypenoside Xvii NA 250000 NA NA NA NA TTD
TOP1 Ginsenoside-F5 NA 250000 NA NA NA NA TTD
TOP1 2, 3-Dihydroxy-12-ursen-28-oic acid NA 250000 NA NA NA NA TTD