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      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TOP1 Ginsenoside F3 NA 250000 NA NA NA NA TTD
TOP1 20(R)-Ginsenoside Rg2 NA 250000 NA NA NA NA TTD
TOP1 (20R)-Ginsenoside Rg3 NA 250000 NA NA NA NA TTD
TOP1 Quasipanaxatriol NA 250000 NA NA NA NA TTD
TOP1 [(3R,4R,4aR,5R,6aR,6aS,6bR,8aR,9S,10S,12aR,14bS)-5,10-dihydroxy-4a,9-bis(hydroxymethyl)-2,2,6a,6b,9,12a-hexamethyl-4-[(Z)-2-methylbut-2-enoyl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-3-yl] (Z)-2-methylbut-2-enoate NA 250000 NA NA NA NA TTD
TOP1 [(3R,4R,4aR,5S,6R,6aR,6aS,6bR,8aR,10S,12aR,14bS)-5,6,10-trihydroxy-4a-(hydroxymethyl)-2,2,6a,6b,9,9,12a-heptamethyl-3-[(Z)-2-methylbut-2-enoyl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4-yl] 2-methylbutanoate NA 250000 NA NA NA NA TTD
TOP1 [(3R,4R,4aR,5R,6aR,6aS,6bR,8aR,10S,12aR,14bS)-5,10-dihydroxy-4a-(hydroxymethyl)-2,2,6a,6b,9,9,12a-heptamethyl-3-[(Z)-2-methylbut-2-enoyl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-4-yl] 2-methylbutanoate NA 250000 NA NA NA NA TTD
TOP1 [(3R,4R,4aR,5R,6aR,6aS,6bR,8aR,9S,10S,12aR,14bS)-5,10-dihydroxy-4a,9-bis(hydroxymethyl)-2,2,6a,6b,9,12a-hexamethyl-4-(2-methylpropanoyloxy)-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicen-3-yl] (Z)-2-methylbut-2-enoate NA 250000 NA NA NA NA TTD
TOP1 Aesculioside IIi NA 250000 NA NA NA NA TTD
TOP1 Eryngiioside J NA 250000 NA NA NA NA TTD
TOP1 Saniculasaponin III NA 250000 NA NA NA NA TTD
TOP1 Eryngiioside L NA 250000 NA NA NA NA TTD
TOP1 Aesculioside IIg NA 250000 NA NA NA NA TTD
TOP1 Aesculioside IIk NA 250000 NA NA NA NA TTD
TOP1 Aesculioside IIa NA 109300 NA NA NA NA TTD
TOP1 Eryngioside 94A NA 250000 NA NA NA NA TTD
TOP1 21-Angeloyl-protoaescigenin NA 250000 NA NA NA NA TTD
TOP1 Eryngioside F NA 250000 NA NA NA NA TTD
TOP1 Eryngioside E NA 250000 NA NA NA NA TTD
TOP1 Aesculioside IIj NA 250000 NA NA NA NA TTD