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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TP53 1-(9-ethyl-9H-carbazol-3-yl)-N-methylmethanamine NA NA 140000 NA NA NA BindingDB
TP53 Propofol NA NA NA NA 108707 NA PubChem
TP53 2-Phenylphenol NA NA NA NA 446684 NA PubChem
TP53 3,5-Diiodosalicylic acid NA NA 820000 NA NA NA BindingDB
TP53 Miristalkonium chloride NA NA NA NA 2511890 NA PubChem
TPH1 US10214530, Example 34 NA 206000 NA NA NA NA BindingDB
TPH1 US10683309, Example 24 NA 133600 NA NA NA NA BindingDB
TPMT Vanillic Acid NA 478630 NA NA NA NA PubChem
TPMT 4-Aminobenzoic Acid NA 2884030 NA NA NA NA PubChem
TPSAB1 Piperazine-1,4-dicarboxylic acid ethylamide 4-guanidino-benzylamide 370000 NA NA NA NA NA TTD
TPSAB1 [5-[4-(Benzylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(benzylcarbamoyl)piperazine-1-carboxylate 101000 NA NA NA NA NA TTD
TPSAB1 (R)-2-Acetylamino-3-(4-aminomethyl-phenyl)-propionic acid methyl ester 213000 NA NA NA NA NA TTD
TPSB2 2-Aminoquinoline 220000 NA NA NA NA NA BindingDB
TPSB2 2-Aminobenzimidazole 110000 NA NA NA NA NA BindingDB
TPSB2 2-(pyridin-2-ylmethyl)-1H-benzimidazole-6-carboximidamide 358000 NA NA NA NA NA BindingDB
TPSB2 Piperazine-1,4-dicarboxylic acid ethylamide 4-guanidino-benzylamide 370000 NA NA NA NA NA BindingDB
TPSB2 [5-[4-[2-(1-Ethanimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-ethanimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carboxylate 255000 NA NA NA NA NA BindingDB
TPSB2 [5-[4-(Benzylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(benzylcarbamoyl)piperazine-1-carboxylate 101000 NA NA NA NA NA BindingDB
TPSB2 (R)-2-Acetylamino-3-(4-aminomethyl-phenyl)-propionic acid methyl ester 213000 NA NA NA NA NA BindingDB
TPSB2 2,4-Diaminoquinazoline 1200000 NA NA NA NA NA BindingDB