GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
TRPA1 |
2-{[(2E)-3-(4-nitrophenyl)prop-2-enoyl]amino}benzoic acid |
NA |
NA |
NA |
199526.23 |
NA |
NA |
TTD |
TRPA1 |
1,7,7-Trimethylbicyclo[2.2.1]heptan-2-ol |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
TRPA1 |
Borneol |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
TRPA1 |
2-Chlorophenol |
NA |
NA |
NA |
501000 |
NA |
NA |
PubChem |
TRPA1 |
Isoeugenol |
NA |
NA |
NA |
149000 |
NA |
NA |
PubChem |
TRPA1 |
Nicotine |
NA |
NA |
NA |
457088000 |
NA |
NA |
PubChem |
TRPM2 |
8-Bromoadenosine 5'-diphosphoribose |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
TRPM2 |
Mefenamic Acid |
NA |
124000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
TRPM2 |
Niflumic Acid |
NA |
149000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
TRPM3 |
Halothane |
NA |
520000 |
NA |
NA |
NA |
NA |
GtoPDB |
TRPM3 |
Chloroform |
NA |
167000 |
NA |
NA |
NA |
NA |
GtoPDB |
TRPM4 |
Adenosine |
NA |
630000 |
NA |
NA |
NA |
NA |
GtoPDB |
TRPM7 |
Nafamostat |
NA |
617000 |
NA |
NA |
NA |
NA |
GtoPDB |
TRPM8 |
Menthol |
NA |
NA|520000 |
NA |
818000|NA |
NA |
NA |
PubChem |
TRPM8 |
Geraniol |
NA |
NA |
NA |
5900000 |
NA |
NA |
PubChem|TTD |
TRPV1 |
N-3,7-Dimethyl-2,6-octadienyl cyclopropylcarboxamide, (2E)- |
NA |
NA |
NA |
115000 |
NA |
NA |
BindingDB|TTD |
TRPV1 |
methyl (1S,14R,16S,17S)-16-ethyl-7-methoxy-3-(methoxymethyl)-10,12-diazapentacyclo[12.3.1.02,10.04,9.012,17]octadeca-2,4(9),5,7-tetraene-1-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
TRPV1 |
[2-[2-(5-hydroxy-1H-indol-3-yl)ethylcarbamoyl]phenyl] acetate |
NA |
203000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
TRPV1 |
[(1S,15R,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-1-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
TRPV1 |
2-Aminoethoxydiphenylborate |
NA |
NA |
NA |
129000 |
NA |
NA |
BindingDB|TTD |