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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TRPA1 2-{[(2E)-3-(4-nitrophenyl)prop-2-enoyl]amino}benzoic acid NA NA NA 199526.23 NA NA TTD
TRPA1 1,7,7-Trimethylbicyclo[2.2.1]heptan-2-ol NA 300000 NA NA NA NA PubChem
TRPA1 Borneol NA 300000 NA NA NA NA TTD
TRPA1 2-Chlorophenol NA NA NA 501000 NA NA PubChem
TRPA1 Isoeugenol NA NA NA 149000 NA NA PubChem
TRPA1 Nicotine NA NA NA 457088000 NA NA PubChem
TRPM2 8-Bromoadenosine 5'-diphosphoribose NA 300000 NA NA NA NA BindingDB|TTD
TRPM2 Mefenamic Acid NA 124000 NA NA NA NA PubChem|TTD
TRPM2 Niflumic Acid NA 149000 NA NA NA NA PubChem|TTD
TRPM3 Halothane NA 520000 NA NA NA NA GtoPDB
TRPM3 Chloroform NA 167000 NA NA NA NA GtoPDB
TRPM4 Adenosine NA 630000 NA NA NA NA GtoPDB
TRPM7 Nafamostat NA 617000 NA NA NA NA GtoPDB
TRPM8 Menthol NA NA|520000 NA 818000|NA NA NA PubChem
TRPM8 Geraniol NA NA NA 5900000 NA NA PubChem|TTD
TRPV1 N-3,7-Dimethyl-2,6-octadienyl cyclopropylcarboxamide, (2E)- NA NA NA 115000 NA NA BindingDB|TTD
TRPV1 methyl (1S,14R,16S,17S)-16-ethyl-7-methoxy-3-(methoxymethyl)-10,12-diazapentacyclo[12.3.1.02,10.04,9.012,17]octadeca-2,4(9),5,7-tetraene-1-carboxylate NA 200000 NA NA NA NA TTD
TRPV1 [2-[2-(5-hydroxy-1H-indol-3-yl)ethylcarbamoyl]phenyl] acetate NA 203000 NA NA NA NA BindingDB|TTD
TRPV1 [(1S,15R,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-1-yl]methanol NA 200000 NA NA NA NA BindingDB|TTD
TRPV1 2-Aminoethoxydiphenylborate NA NA NA 129000 NA NA BindingDB|TTD