| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TRPV1 |
4-Hydroxybenzyl isothiocyanate |
NA |
NA |
NA |
170000 |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
Phenethyl Isothiocyanate |
NA |
NA |
NA |
180000 |
NA |
NA |
BindingDB|PubChem|TTD |
| TRPV1 |
(4-Hydroxy-3-methoxyphenyl)methyl 3-[4-[(3,5-difluorophenyl)sulfonylamino]-3,5-dihydroxyphenyl]propanoate |
NA |
NA |
273200 |
NA |
NA |
NA |
BindingDB |
| TRPV1 |
N-[beta-(3,4-Dihydroxyphenyl)-ethyl]-2,2-dimethylpropionamide |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| TRPV1 |
methyl (1S,10S,15R,17S,18S)-17-ethyl-10-hydroxy-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1-carboxylate |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
Benzyl Isothiocyanate |
NA |
NA |
NA |
223000 |
NA |
NA |
BindingDB|PubChem|TTD |
| TRPV1 |
19(S)-Heyneanine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| TRPV1 |
Nobilamide B |
NA |
275000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
Nobilamide A |
NA |
1665000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
(R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-isopropyl-6,13-dimethyl-2,5,8,11-tetraoxo-1-oxa-4,7,10-triazacyclotridecan-12-ylamino)-1-oxo-3-phenylpropan-2-yl)-4-methylpentanamide |
NA |
1320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
(R)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-isopropyl-6,13-dimethyl-2,5,8,11-tetraoxo-1-oxa-4,7,10-triazacyclotridecan-12-ylamino)-1-oxo-3-phenylpropan-2-yl)-4-methyl-2-((R)-3-phenyl-2-propionamidopropanamido)pentanamide |
NA |
227000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV1 |
Allyl Isothiocyanate |
NA |
NA |
NA |
160000 |
NA |
NA |
BindingDB|PubChem|TTD |
| TRPV1 |
Cannabidiol |
NA |
NA |
110400 |
NA |
NA |
NA |
BindingDB |
| TRPV1 |
Coronaridine |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV3 |
Cannabichromene |
NA |
201000 |
NA |
NA |
NA |
NA |
BindingDB |
| TRPV4 |
Vildagliptin |
NA |
NA |
NA |
1000000 |
NA |
NA |
GtoPDB |
| TRPV4 |
4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide |
NA |
NA |
NA |
125892.54 |
NA |
NA |
TTD |
| TRPV6 |
11-Hydroxy-5,6-dihydrobenzo[b][1]benzoborepine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| TRPV6 |
2-Benzhydryloxyethanamine |
NA |
159100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| TRPV6 |
2,2-Diphenyl-1-thia-3-azonia-2-boranuidacyclopentane |
NA |
127100 |
NA |
NA |
NA |
NA |
BindingDB |