Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
TPSB2 | 1-Aminoisoquinoline | 390000 | NA | NA | NA | NA | NA | BindingDB |
TPSB2 | 1H-Benzimidazol-2-amine, 1-methyl- | 1800000 | NA | NA | NA | NA | NA | BindingDB |
TPSB2 | 5,6-Dimethylbenzimidazol-2-ylamine | 220000 | NA | NA | NA | NA | NA | BindingDB |
TPST2 | NA | 425000 | NA | NA | NA | NA | BindingDB | |
TRAP1 | 8-((3,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine | NA | 157900 | NA | NA | NA | NA | BindingDB |
TRAP1 | 8-((2,4-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine | NA | 145400 | NA | NA | NA | NA | BindingDB |
TRAP1 | 8-((2,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine | NA | 203700 | NA | NA | NA | NA | BindingDB |
TREH | 2-Butyl-6-hydroxymethyl-piperidine-3,4,5-triol | NA | 780000 | NA | NA | NA | NA | BindingDB |
TRPA1 | Allyl Sulfide | NA | NA | NA | 254000 | NA | NA | PubChem|TTD |
TRPA1 | 2-[[(E)-3-(4-methylphenyl)prop-2-enoyl]amino]benzoic acid | NA | NA | NA | 149000 | NA | NA | TTD |
TRPA1 | (6S)-6-[3-(3-methoxypropoxy)phenyl]-8-oxa-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene-4-thione | NA | 40000000 | NA | NA | NA | NA | TTD |
TRPA1 | Urb-597 | NA | NA | NA | 134896000 | NA | NA | PubChem |
TRPA1 | Camphor (synthetic) | NA | 660000|400000 | NA | NA | NA | NA | PubChem|TTD |
TRPA1 | 2-{[(2E)-2-methyl-3-phenylprop-2-enoyl]amino}benzoic acid | NA | NA | NA | 125892.54 | NA | NA | TTD |
TRPA1 | Diclofenac | NA | NA | NA | 210000 | NA | NA | PubChem |
TRPA1 | Eugenol | NA | NA | NA | 168000|169824|116000|261000 | NA | NA | PubChem|TTD |
TRPA1 | Iodoacetamide | NA | NA | NA | 357000 | NA | NA | TTD |
TRPA1 | N-Hex-5-ynyl-2-iodo-acetamide | NA | NA | NA | 134000 | NA | NA | TTD |
TRPA1 | Probenecid | NA | NA | NA | 4200000 | NA | NA | PubChem|TTD |
TRPA1 | Tranilast | NA | 125893|126000|125892.54 | NA | NA | NA | NA | PubChem|TTD |