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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
TPSB2 1-Aminoisoquinoline 390000 NA NA NA NA NA BindingDB
TPSB2 1H-Benzimidazol-2-amine, 1-methyl- 1800000 NA NA NA NA NA BindingDB
TPSB2 5,6-Dimethylbenzimidazol-2-ylamine 220000 NA NA NA NA NA BindingDB
TPST2 NA 425000 NA NA NA NA BindingDB
TRAP1 8-((3,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine NA 157900 NA NA NA NA BindingDB
TRAP1 8-((2,4-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine NA 145400 NA NA NA NA BindingDB
TRAP1 8-((2,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amine NA 203700 NA NA NA NA BindingDB
TREH 2-Butyl-6-hydroxymethyl-piperidine-3,4,5-triol NA 780000 NA NA NA NA BindingDB
TRPA1 Allyl Sulfide NA NA NA 254000 NA NA PubChem|TTD
TRPA1 2-[[(E)-3-(4-methylphenyl)prop-2-enoyl]amino]benzoic acid NA NA NA 149000 NA NA TTD
TRPA1 (6S)-6-[3-(3-methoxypropoxy)phenyl]-8-oxa-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene-4-thione NA 40000000 NA NA NA NA TTD
TRPA1 Urb-597 NA NA NA 134896000 NA NA PubChem
TRPA1 Camphor (synthetic) NA 660000|400000 NA NA NA NA PubChem|TTD
TRPA1 2-{[(2E)-2-methyl-3-phenylprop-2-enoyl]amino}benzoic acid NA NA NA 125892.54 NA NA TTD
TRPA1 Diclofenac NA NA NA 210000 NA NA PubChem
TRPA1 Eugenol NA NA NA 168000|169824|116000|261000 NA NA PubChem|TTD
TRPA1 Iodoacetamide NA NA NA 357000 NA NA TTD
TRPA1 N-Hex-5-ynyl-2-iodo-acetamide NA NA NA 134000 NA NA TTD
TRPA1 Probenecid NA NA NA 4200000 NA NA PubChem|TTD
TRPA1 Tranilast NA 125893|126000|125892.54 NA NA NA NA PubChem|TTD