| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| TSPO |
7-bromo-5-(2,6-difluorophenyl)-1-methyl-3H-1,4-benzodiazepin-2-one |
NA |
416869383.5 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
2H-1,4-Benzodiazepin-2-one, 5-(2-fluorophenyl)-1,3-dihydro-7-(hydroxyamino)-1-methyl- |
NA |
10423174.29 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
1,3-Dihydro-7-nitro-5-(alpha,alpha,alpha-trifluoro-o-tolyl)2H-1,4-benzodiazepin-2-one |
NA |
285759054.3 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-5-phenyl-7-(trifluoromethyl)- |
NA |
76913044.03 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
Delorazepam |
NA |
555904000|555904257.3 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TSPO |
7-Aminoclonazepam |
NA |
13335214.32 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
1H-1,4-Benzodiazepine-7-carbonitrile, 2,3-dihydro-1-methyl-2-oxo-5-phenyl- |
NA |
2630267.99 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
5-(2-Fluorophenyl)-1,3-dihydro-1-methyl-2H-1,4-benzodiazepin-2-one |
NA |
71449632.61 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
5-(o-fluorophenyl)-2,3-dihydro-1-methyl-2-oxo-1H-1,4-benzodiazepine-7-carbonitrile |
NA |
33342641.28 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
7-Amino Nimetazepam |
NA |
2172701.18 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
1-Methyl-5-(2-fluorophenyl)-7-fluoro-1,3-dihydro-2h-1,4-benzodiazepine-2-one |
NA |
195884467.4 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
1,4-Benzdiazepin-2-one-5(26F-PH)8CL |
NA |
35727283.82 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
7-Chloro-5-(2,6-difluorophenyl)-1,3-dihydro-2H-1,4-benzodiazepin-2-one |
NA |
625172692.8 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
7-acetyl-5-(o-fluorophenyl)-1,3-dihydro-2H-1,4-benzodiazepin-2-one |
NA |
55590425.73 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
Clonazepam |
NA |
555904000|555904257.3 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TSPO |
Nordazepam |
NA |
106414000|106414301.8 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TSPO |
Diazepam |
NA |
123595000|123594743.3 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TSPO |
2H-1,4-Benzodiazepin-2-one, 1,3-dihydro-7-chloro-5-(2-fluorophenyl)-1-(2-hydroxyethyl)- |
NA |
40831938.63 |
NA |
NA |
NA |
NA |
TTD |
| TSPO |
Halazepam |
NA |
10864300|10864256.24 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| TSPO |
Flunitrazepam |
NA |
263027000|263026799.2 |
NA |
NA |
NA |
NA |
PubChem|TTD |