| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ADORA3 |
4-(Furan-2-yl)-11-(2-phenylethyl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-amine |
281838.29 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
6,7-dimethoxy-4H-indeno[1,2-d][1,3]thiazol-2-amine;hydroiodide |
NA |
NA |
NA |
794328|794328.23 |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
|
346736.85 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
N-(3-pyridin-2-ylisoquinolin-1-yl)benzamide |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
179999 |
PubChem |
| ADORA3 |
1-(2-Phenyl-quinazolin-4-yl)-3-o-tolyl-urea |
115000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
N-(2,6-Dimethyl-benzoyl)-2,6-dimethyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benzamide |
3200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
N-(3-Pyridin-2-yl-isoquinolin-1-yl)-formamidine |
20000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
N-Benzoyl-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benzamide |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
1-Phenyl-3-(quinazolin-4-yl)urea |
1180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-Phenyl-3-(2-phenyl-quinazolin-4-yl)-urea |
287000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
3,4-dimethoxy-N-(3-(pyridin-2-yl)isoquinolin-1-yl)benzamide |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine |
301995.17 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-(2-tert-Butyl-quinazolin-4-yl)-3-phenyl-urea |
78700000 |
NA |
NA |
NA |
NA|NA |
NA|NA |
BindingDB|TTD |
| ADORA3 |
8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine |
602559.59 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-ethanone |
660000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-(2-(Diethylamino)quinazolin-4-yl)-3-phenylurea |
178000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-[2-(4,6-Dimethyl-pyrimidin-2-yl)-quinazolin-4-yl]-3-phenyl-urea |
1260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
5-Amino-8-ethyl-2-(2-furyl)-pyrazolo[4,3-e] 1,2,4-triazolo[1,5-c]pyrimidine |
407380.28 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
11-Tert-butyl-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-amine |
1148153.62 |
NA |
NA |
NA |
NA |
NA |
BindingDB |