| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ADORA3 |
[4-(1,4-dioxo-5H-[1,2,4]triazolo[4,3-a]quinoxalin-2-yl)phenyl] acetate |
4950000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
11-(Cyclohexylmethyl)-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-amine |
1737800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-Amino-2-(4-ethoxy-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
3690000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-Amino-2-(4-amino-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
3470000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
6-Amino-2-(4-methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]quinoxaline-1,4-dione |
4080000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4,6-Diamino-2-(4-methoxy-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
4650000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
2-(4-Dimethylamino-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]quinoxaline-1,4-dione |
3360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-Amino-2-(4-hydroxy-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
4130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
2-(4-methoxyphenyl)-6-nitro-[1,2,4]triazolo[4,3-a]quinoxaline-1,4(2H,5H)-dione |
5330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4,6-Diamino-2-(4-hydroxy-phenyl)-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
3570000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-(Furan-2-yl)-11-octyl-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-amine |
2041737.94 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-Amino-6-nitro-2-phenyl-2H-[1,2,4]triazolo[4,3-a]quinoxalin-1-one |
5320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
4-amino-2-(4-methoxyphenyl)-6-nitro-[1,2,4]triazolo[4,3-a]quinoxalin-1(2H)-one |
4330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
1-Methoxy-3-pyridin-2-yl-isoquinoline |
5600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
N-(2-Pyridin-2-yl-quinazolin-4-yl)-benzamide |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
N-Benzoyl-N-(2-pyridin-2-yl-quinazolin-4-yl)-benzamide |
470000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
2,2,2-Trifluoro-N-(2-pyridin-2-yl-quinazolin-4-yl)-acetamide |
86000000 |
NA |
NA |
NA |
NA|NA |
NA|NA |
BindingDB|TTD |
| ADORA3 |
N-(2-Pyridin-2-yl-quinazolin-4-yl)-formamidine |
4000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
1-Ethyl-3-pyridin-2-yl-isoquinoline |
5100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
4-Hydroxy-2-(2-pyridyl)quinazoline |
22000000 |
NA |
NA |
NA |
NA |
NA |
TTD |