Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ADORA3 N-(2-Pyridin-2-yl-quinazolin-4-yl)-acetamide 11000000 NA NA NA NA NA BindingDB|TTD
ADORA3 Meropenem NA NA NA NA NA 300000 PubChem
ADORA3 3-Chloro-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benzamidine 7800000 NA NA NA NA NA BindingDB|TTD
ADORA3 4-Chloro-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benzamidine 2300000 NA NA NA NA NA BindingDB|TTD
ADORA3 tert-butyl N-[4-[[4-(furan-2-yl)-11-(2-phenylethyl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-yl]amino]-4-oxobutyl]carbamate 1479108.39 NA NA NA NA NA BindingDB
ADORA3 tert-butyl N-[4-[[4-(furan-2-yl)-11-(3-methylbutyl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(12),2,4,7,9-pentaen-7-yl]amino]-4-oxobutyl]carbamate 2511886.43 NA NA NA NA NA BindingDB
ADORA3 2'-Amino-2'-deoxyadenosine 1000000 NA NA NA NA NA BindingDB
ADORA3 5'-N-Ethylcarboxamidoadenosine NA NA NA 303000 NA NA BindingDB
ADORA3 3-methyl-N-[3-(2-pyridyl)-1-isoquinolyl]benzamidine 1300000 NA NA NA NA NA BindingDB|TTD
ADORA3 3,4-dichloro-N-[3-(2-pyridyl)-1-isoquinolyl]benzamidine 2300000 NA NA NA NA NA BindingDB|TTD
ADORA3 N-[3-(2-pyridyl)-1-isoquinolyl]benzamidine 740000 NA NA NA NA NA BindingDB
ADORA3 [(4-Methoxyphenyl)iminomethyl](3-(2-pyridyl)isoquinolyl)amine 310000 NA NA NA NA NA BindingDB|TTD
ADORA3 3-methoxy-N-[3-(2-pyridyl)-1-isoquinolyl]benzamidine 980000 NA NA NA NA NA BindingDB|TTD
ADORA3 N-(3-Pyridin-2-yl-isoquinolin-1-yl)-isobutyramide 48000000 NA NA NA NA NA BindingDB|TTD
ADORA3 Theobromine 103000 NA NA NA NA NA BindingDB|PubChem
ADORA3 Cefepime NA NA NA NA NA 300000 PubChem
ADORA3 Ceftazidime NA NA NA NA NA 300000 PubChem
ADORA3 5-Phenyl-1,2,4-thiadiazol-3-amine NA NA 102000 NA NA NA BindingDB|ChEMBL
ADORA3 Aztreonam NA NA NA NA NA 400000 PubChem
ADORA3 1-(Methylthio)-3-pyridin-2-ylisoquinoline 3900000 NA NA NA NA NA BindingDB|TTD