| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ADORA3 |
1-(Methylsulfonyl)-3-pyridin-2-ylisoquinoline |
15000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
N-acetyl-N-(3-pyridin-2-ylisoquinolin-1-yl)acetamide |
35000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| ADORA3 |
|
22000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
2,4-Diamino-6-phenyl-1,3,5-triazine |
NA |
NA |
104200 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| ADORA3 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ADORA3 |
3-Pyridin-2-yl-isoquinolin-1-ol |
27000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
1-Chloro-3-pyridin-2-yl-isoquinoline |
2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylcarbamoyl)-methyl-ammonium; chloride |
162929.6 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
5'-Amino-5'-deoxyadenosine |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADORA3 |
(2-amino-4H-indeno[1,2-d][1,3]thiazol-5-yl) acetate;hydroiodide |
NA |
NA |
NA |
15848932|15848931.92 |
NA |
NA |
BindingDB|TTD |
| ADORA3 |
2-(4-Nitro-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]quinoxaline-1,4-dione |
6220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ADRA1A |
Phenylpropanolamine |
NA |
NA |
NA |
230000 |
NA |
NA |
PubChem |
| ADRA1A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ADRA1A |
4-(2-Amino-1-hydroxyethyl)-5-fluorobenzene-1,2-diol |
NA |
NA |
NA |
125000 |
NA |
NA |
BindingDB |
| ADRA1A |
4-(4,5-Dihydro-1,3-oxazol-2-yl)morpholine |
107152|120226|107151.93 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADRA1A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ADRA1A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ADRA1A |
(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol |
340000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ADRA1A |
(1S,2R)-(+)-Norephedrine |
NA |
NA |
NA |
230000 |
NA |
NA |
BindingDB|TTD |