| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| APH1A |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| APH1A |
9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| APH1A |
2-(9-Octylcarbazol-2-yl)oxyacetamide |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| APH1A |
2-(9-Octylcarbazol-2-yl)oxyacetonitrile |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| APH1A |
4-[4-[(Z)-(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-2-methoxyphenoxy]butanenitrile |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| APH1A |
Tarenflurbil |
NA |
307000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| APH1B |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| APH1B |
9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| APH1B |
2-(9-Octylcarbazol-2-yl)oxyacetamide |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| APH1B |
2-(9-Octylcarbazol-2-yl)oxyacetonitrile |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| APH1B |
4-[4-[(Z)-(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-2-methoxyphenoxy]butanenitrile |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| APH1B |
Tarenflurbil |
NA |
307000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| APLNR |
US11020395, Example 58.0 |
NA |
NA |
NA |
179000 |
NA |
NA |
BindingDB |
| APLNR |
US11020395, Example 64.0 |
NA |
NA |
NA |
146000 |
NA |
NA |
BindingDB |
| APP |
methyl 2,4-dihydroxy-6-methyl-3-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienyl]benzoate |
NA |
221000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
Chf 5022 |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
CID 10529819 |
NA |
NA |
NA |
112600 |
NA |
NA |
BindingDB|TTD |
| APP |
4-Bromo-2-((furan-2-ylmethyl)amino)benzoic acid |
NA |
154420 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
1-[4''-(4,4-Dimethyl-cyclohexyl)-2-fluoro-biphenyl-4-yl]-cyclopropanecarboxylic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
2-(4-Benzo[1,3]dioxol-5-yl-3-fluoro-phenyl)-propionic acid |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |